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Letters in Drug Design & Discovery

最近発刊の雑誌の目次より: Letters in Drug Design & Discovery © Bentham Science Publishers
  • Synthesis, DNA-Binding Ability and Biological Activity of C8 Linked G1 Dendrimer-Pyrrolobenzodiazepine Conjugates as Anticancer Agents
    Letters in Drug Design & Discovery, Vol. 5, No. 7. (October 2008), pp. 424-432.
  • Sesquiterpene Lactones and their Anti-Tumor Activity from the Flowers of Inula Britannica
    Letters in Drug Design & Discovery, Vol. 5, No. 7. (October 2008), pp. 433-436.
  • 3D-QSAR Studies of Various Diaryl Urea Derivatives of Multi-targeted Receptor Tyrosine Kinase Inhibitors: Molecular Field Analysis Approach
    Letters in Drug Design & Discovery, Vol. 5, No. 7. (October 2008), pp. 437-448.
  • 3D-QSAR Analysis on N-Phenylacetanoyl-L-Homoserine Lactones as Inhibitors of Bacterial Quorum Sensing via CoMFA Approach
    Letters in Drug Design & Discovery, Vol. 5, No. 7. (October 2008), pp. 449-453.
  • Synthesis and In Vitro Antiproliferative Activity of Diphenyl(piperidin-4- yl)thioamide Methanol Derivatives
    Letters in Drug Design & Discovery, Vol. 5, No. 7. (October 2008), pp. 454-461.
  • Release of a Poorly Soluble Drug from Cross-Linked -Cyclodextrin-Based Polymer Pellets Prepared via Extrusion/Spheronisation
    Letters in Drug Design & Discovery, Vol. 5, No. 7. (October 2008), pp. 462-470.
  • 96-Well Plate Surface Tension Measurements for Fast Determination of Drug Solubility
    Letters in Drug Design & Discovery, Vol. 5, No. 7. (October 2008), pp. 471-476.
  • New Synthetic Chalcones: Cytotoxic Mannich Bases of 6-(4-Chlorocinnamoyl)-2(3H)-benzoxazolone
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 358-361.
  • A Facile Synthesis of 4-Methylumbelliferyl (13)--D-Pentaglucoside
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 362-363.
    by Huang,
  • Synthesis and Anticancer Evaluation of some Newer 2, 5-Disubstituted-1,3, 4-Oxadiazole Analogues
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 364-368.
  • A Preliminary Assessment of the Structure-Activity Relationship of Benzimidazole-Based Anti-Proliferative Agents
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 369-376.
  • Three-Dimensional Quantitative Structure-Activity Relationships for a Large Series of Potent Antitubercular Agents
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 377-387.
  • Antimicrobial Activities of 7-Aminosterol Squalamine Analogues
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 388-393.
  • Octanol Water Partition Coefficient Determination for Model Steroids Using an HPLC Method
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 394-400.
  • Urease and -Chymotrypsin Inhibitory Effects of Selected Urea Derivatives
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 401-405.
  • Nimesulide Apparent Solubility Enhancement with Natural Cyclodextrins and their Polymers
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 406-415.
    by Joudieh, , Lahiani-Skiba, , Bon, , Ba, , Le Breton, , Skiba,
  • Facile Conversion of FP to TR-FRET Assays using Terbium Chelates:Nuclear Receptor Competitive Binding Assays as Examples
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 416-422.
  • Erratum
    Letters in Drug Design & Discovery, Vol. 5, No. 6. (September 2008), pp. 423-423.
  • QSAR Studies on some Calcium Channel Blockers
    Letters in Drug Design & Discovery, Vol. 5, No. 5. (July 2008), pp. 307-312.
    by Naik, A Mallari, Kumar Satuluri, , Gupta,
  • Synthesis of N-Benzenesulfonylbenzotriazole Derivatives, and Evaluation of their Antimicrobial Activity
    Letters in Drug Design & Discovery, Vol. 5, No. 5. (July 2008), pp. 313-318.
  • Virtual Screening of the Guanylate Monophosphate Kinase (GMPK) Family: Investigating the Rules of Ligand Specificity
    Letters in Drug Design & Discovery, Vol. 5, No. 5. (July 2008), pp. 319-326.
  • Antibacterial Pleuromutilin Derivatives based on Alternate Core Structures:Arigoni and Birch Chemistry Revisited
    Letters in Drug Design & Discovery, Vol. 5, No. 5. (July 2008), pp. 327-331.
  • The Interaction of Titanocene Y with Double-Stranded DNA: A Computational Study
    Letters in Drug Design & Discovery, Vol. 5, No. 5. (July 2008), pp. 332-335.
  • Structure-Activity Relationship Study of 8-amino-2,8-dideoxy- -KDO, a Potent CMP-KDO Synthetase Inhibitor
    Letters in Drug Design & Discovery, Vol. 5, No. 5. (July 2008), pp. 336-339.
  • Discovery of AX8312, an N-alkyl-Gly-boro-Pro Derivative that Accelerates Recovery from Neutropenia in the Mouse
    Letters in Drug Design & Discovery, Vol. 5, No. 5. (July 2008), pp. 340-345.
  • Disodium Phosphate of Novel Pyrazole-Linked Norcantharidin Analogs:Design, Synthesis and their Anticancer Evaluation
    Letters in Drug Design & Discovery, Vol. 5, No. 5. (July 2008), pp. 346-352.
  • Synthesis and Biological Evaluation of a New Series of Benzothiazole-Quinolone Hybrids as Antibacterial Agents
    Letters in Drug Design & Discovery, Vol. 5, No. 5. (July 2008), pp. 353-357.
  • Drug Design Should Involve Consideration of Environmental Risk and Hazard
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 232-235.
  • Design and Synthesis of Carbohydrate Derivatives for Antagonistic Activity at Muscarinic Receptor
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 236-242.
  • Schiff Bases of Istain: Potential Anti-Leishmanial Agents
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 243-249.
  • Synthesis of Medicinally Important N-Trimethylene Dipiperidine Sulfonamides and Carboxamides Containing a Substituted Benzophenone Moiety - An Antibacterial Agents
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 250-260.
  • Synthesis and Anticancer Activity of Phthalimido and Naphthalimido Substituted Dihydropyrimidone Conjugates
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 261-270.
  • Selective Androgen Receptor Modulators Antagonize Apolipoprotein E4-Induced Cognitive Impairments
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 271-276.
  • Antimalarial Activity of 2,4-Diaminopyrimidines
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 277-280.
  • A Quantitative Structure-Activity Relationship Study on a Novel Series of Hydroxamic Acid Analogs Acting as Matrix Metalloproteinase Inhibitors
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 281-285.
    by Gupta, , Bagaria, Priyanka, Kumar Satuluri,
  • Synthesis of 5-Arylidene Barbiturates: A Novel Class of DPPH Radical Scavengers
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 286-291.
  • Phenylpyazoleanilides as Potent Inhibitor of IL-15 Dependent T Cell Proliferation. Part 2: Discovery of a New Drug Candidate, Y-320
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 292-296.
  • Modulation by Dopaminergic System of Morphine Withdrawal: In Vitro Evidences
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 297-301.
    by Capasso,
  • A Novel Strategy to Manage Tolerance to Lamotrigine in Bipolar II Depression
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 302-302.
    by Sharma, , Corpse,
  • Tetrahydroisoquinoline-Related Modulators of Multidrug Resistance in Cancer
    Letters in Drug Design & Discovery, Vol. 5, No. 4. (June 2008), pp. 303-306.
    by Li, Yu, Zhang, B Hui, Huang, Wen, Zhen, Xia, Li, Yun
  • Microwaves-Assisted Syntheses of Imidazolylbenzamides and their Antioxidant Activities
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 152-157.
  • Natural Products Biological Screening and Ligand-Based Virtual Screening for the Discovery of New Antileishmanial Agents
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 158-161.
  • Determination of Molecular Properties Effectuating the Growth Inhibition of Mycobacterium Tuberculosis by Various Small Molecule Hydrazides
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 162-168.
  • New 3-Aminosteroid Derivatives as a New Family of Topical Antibacterial Agents Active against Methicillin-Resistant Staphylococcus aureus (MRSA)
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 169-172.
  • A QSAR Study on some Series of ATP-Sensitive Potassium Channel Openers
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 173-177.
    by Kumar Satuluri, , Gupta,
  • Synthesis and Antimalarial Activity of Novel Hydroxyethylamines,Potential Aspartyl Protease Inhibitors
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 178-181.
  • Estrogen Receptor: Structural Differences and Potential Implications on Selectivity Examined by the GRID/CPCA Approach
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 182-192.
    by De Menezes, , Leitao, , Montanari,
  • Inherent Gene Expression Variabilities and the Need for Personalized Drug Dosage
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 193-208.
  • Intravenous Thrombolysis with rt-PA in Acute Stroke Patients Aged 80 Years
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 209-213.
    by Lorenzano, , Orzi, , Puca, , Toni,
  • Synthesis and Biological Evaluation of a Series of 2-(3,4,5-Trimethoxybenzoyl)-Indol-3-yl Acetic Acid Derivatives as Potential Agents against Human Leukemia K562 Cells
    Letters in Drug Design & Discovery, Vol. 5, No. 3. (April 2008), pp. 214-220.
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